4-Amino-3-nitrophenylboronic acid pinacol ester - PMC

Silke Kayser, Jacob C. Hansen, Markus Staudt, Aleksandra Moroz, Younes Larsen, Piero Temperini, Feng Yi, Jed T. Syrenne, Niels Krogsgaard-Larsen, Stylianos Iliadis, Birgitte Nielsen, Kasper B. Hansen, Darryl S. Pickering, Lennart Bunch

ACS Chem Neurosci. Author manuscript; available in PMC 2021 Mar 4.

Published in final edited form as: ACS Chem Neurosci. 2020 Mar 4; 11(5): 674–701. Published online 2020 Feb 17. doi: 10.1021/acschemneuro.0c00003

PMCID:: PMC7227796

Abstract Article PDF–2.7M

Select item 114348956.

Approachable Synthetic Methodologies for Second-Generation β-Lactamase Inhibitors: A Review

Noor Fatima, Shehla Khalid, Nasir Rasool, Muhammad Imran, Bushra Parveen, Aqsa Kanwal, Marius Irimie, Codrut Ioan Ciurea

Pharmaceuticals (Basel) 2024 Sep; 17(9): 1108. Published online 2024 Aug 23. doi: 10.3390/ph17091108

PMCID:: PMC11434895

Abstract Article PDF–15M

Select item 28796487.

Copper(II)-Catalyzed Conversion of Aryl/Heteroaryl Boronic Acids, Boronates, and Trifluoroborates into the Corresponding Azides: Substrate Scope and Limitations

Kimberly D. Grimes, Amol Gupte, Courtney C. Aldrich

Synthesis (Stuttg) Author manuscript; available in PMC 2010 Nov 1.

Published in final edited form as: Synthesis (Stuttg). 2010 May 1; 2010(9): 1441–1448. doi: 10.1055/s-0029-1218683

PMCID:: PMC2879648

Abstract Article PDF–330K

Select item 75459538.

Boronate-Based Probes for Biological Oxidants: A Novel Class of Molecular Tools for Redox Biology

Adam Sikora, Jacek Zielonka, Karolina Dębowska, Radosław Michalski, Renata Smulik-Izydorczyk, Jakub Pięta, Radosław Podsiadły, Angelika Artelska, Karolina Pierzchała, Balaraman Kalyanaraman

Front Chem. 2020; 8: 580899. Published online 2020 Sep 25. doi: 10.3389/fchem.2020.580899

PMCID:: PMC7545953

Abstract Article PDF–4.0M

Select item 74606369.

Synthesis and Pharmacological Characterization of 2-Aminoethyl Diphenylborinate (2-APB) Derivatives for Inhibition of Store-Operated Calcium Entry (SOCE) in MDA-MB-231 Breast Cancer Cells

Achille Schild, Rajesh Bhardwaj, Nicolas Wenger, Dominic Tscherrig, Palanivel Kandasamy, Jan Dernič, Roland Baur, Christine Peinelt, Matthias A. Hediger, Martin Lochner

Int J Mol Sci. 2020 Aug; 21(16): 5604. Published online 2020 Aug 5. doi: 10.3390/ijms21165604

PMCID:: PMC7460636

Abstract Article PDF–5.5M

Select item 313414110.

Suzuki–Miyaura cross-coupling reaction on copper-trans-A₂B corroles with excellent functional group tolerance

Michael König, Lorenz Michael Reith, Uwe Monkowius, Günther Knör, Klaus Bretterbauer, Wolfgang Schoefberger

Tetrahedron. 2011 Jun 10; 67(23): 4243–4252. doi: 10.1016/j.tet.2011.04.024

PMCID:: PMC3134141

Abstract Article

Select item 930268711.

Nickel‐Catalyzed Arylative Cyclizations of Alkyne‐ and Allene‐Tethered Electrophiles using Arylboron Reagents

Simone M. Gillbard, Prof. Hon Wai Lam

Chemistry. 2022 Mar 28; 28(18): e202104230. Published online 2022 Jan 27. doi: 10.1002/chem.202104230

PMCID:: PMC9302687

Abstract Article PDF–18M

Select item 981797012.

Identification of Thiazolo[5,4-b]pyridine Derivatives as c-KIT Inhibitors for Overcoming Imatinib Resistance

Yunju Nam, Chan Kim, Junghee Han, SeongShick Ryu, Hanna Cho, Chiman Song, Nam Doo Kim, Namkyoung Kim, Taebo Sim

Cancers (Basel) 2023 Jan; 15(1): 143. Published online 2022 Dec 26. doi: 10.3390/cancers15010143

Correction in:: Cancers (Basel). 2024 Jun; 16(11): 2151.

PMCID:: PMC9817970

Abstract Article PDF–18M

Select item 563259613.

Extremely long tumor retention, multi-responsive boronate crosslinked micelles with superior therapeutic efficacy for ovarian cancer

Wenwu Xiao, Nell Suby, Kai Xiao, Tzu-yin Lin, Nasir Al Awwad, Kit S. Lam, Yuanpei Li

J Control Release. Author manuscript; available in PMC 2018 Oct 28.

Published in final edited form as: J Control Release. 2017 Oct 28; 264: 169–179. Published online 2017 Aug 25. doi: 10.1016/j.jconrel.2017.08.028

PMCID:: PMC5632596

Abstract Article PDF–3.7M

Select item 889012714.

Exponential amplification by redox cross-catalysis and unmasking of doubly protected molecular probes

Justine Pallu, Charlie Rabin, Pan Hui, Thamires S. Moreira, Geordie Creste, Corentin Calvet, Benoît Limoges, François Mavré, Mathieu Branca

Chem Sci. 2022 Mar 2; 13(9): 2764–2777. Published online 2022 Feb 11. doi: 10.1039/d1sc06086d

PMCID:: PMC8890127

Abstract Article PDF–1.6M

Select item 918636215.

Design and biological evaluation of substituted 5,7-dihydro-6H-indolo[2,3-c]quinolin-6-one as novel selective Haspin inhibitors

Sreenivas Avula, Xudan Peng, Xingfen Lang, Micky Tortorella, Béatrice Josselin, Stéphane Bach, Stephane Bourg, Pascal Bonnet, Frédéric Buron, Sandrine Ruchaud, Sylvain Routier, Cleopatra Neagoie

J Enzyme Inhib Med Chem. 2022; 37(1): 1632–1650. Published online 2022 Jun 7. doi: 10.1080/14756366.2022.2082419

PMCID:: PMC9186362

Abstract Article PDF–4.5M

Select item 725307616.

Development of MAP4 kinase inhibitors as motor-neuron-protecting agents

Pieter H. Bos, Emily R. Lowry, Jonathon Costa, Sebastian Thams, Alejandro Garcia-Diaz, Arie Zask, Hynek Wichterle, Brent R. Stockwell

Cell Chem Biol. Author manuscript; available in PMC 2020 Dec 19.

Published in final edited form as: Cell Chem Biol. 2019 Dec 19; 26(12): 1703–1715.e37. Published online 2019 Oct 31. doi: 10.1016/j.chembiol.2019.10.005