3-Bromo-5-(trifluoromethyl)phenylboronic acid - PMC

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Items: 12

Select item 72487031.

Efficient Access to 3,5-Disubstituted 7-(Trifluoromethyl)pyrazolo[1,5-a]pyrimidines Involving S_NAr and Suzuki Cross-Coupling Reactions

Badr Jismy, Abdellatif Tikad, Mohamed Akssira, Gérald Guillaumet, Mohamed Abarbri

Molecules. 2020 May; 25(9): 2062. Published online 2020 Apr 28. doi: 10.3390/molecules25092062

PMCID:: PMC7248703

Abstract Article PDF–1.2M

Select item 104612302.

Inhibition of FLT3-ITD Kinase in Acute Myeloid Leukemia by New Imidazo[1,2-b]pyridazine Derivatives Identified by Scaffold Hopping

Petra Břehová, Eva Řezníčková, Kryštof Škach, Radek Jorda, Milan Dejmek, Veronika Vojáčková, Michal Šála, Markéta Kovalová, Martin Dračínský, Alexandra Dolníková, Timotej Strmeň, Monika Kinnertová, Karel Chalupský, Alexandra Dvořáková, Tomáš Gucký, Helena Mertlíková Kaiserová, Pavel Klener, Radim Nencka, Vladimír Kryštof

J Med Chem. 2023 Aug 24; 66(16): 11133–11157. Published online 2023 Aug 3. doi: 10.1021/acs.jmedchem.3c00575

PMCID:: PMC10461230

Abstract Article PDF–7.7M

Select item 107138513.

Base-assisted transmetalation enables gold-catalyzed oxidative Sonogashira coupling reaction

Lizhu Zhang, Wenchao Zhang, Dinghua Li, Rongjie Yang, Zhonghua Xia

iScience. 2024 Jan 19; 27(1): 108531. Published online 2023 Nov 23. doi: 10.1016/j.isci.2023.108531

PMCID:: PMC10713851

Abstract Article PDF–8.6M

Select item 59652594.

Species-Selective Pyrimidineamine Inhibitors of Trypanosoma brucei S-Adenosylmethionine Decarboxylase

Oleg A. Volkov, Anthony J. Brockway, Stephen A. Wring, Michael Peel, Zhe Chen, Margaret A. Phillips, Jef K. De Brabander

J Med Chem. Author manuscript; available in PMC 2019 Feb 8.

Published in final edited form as: J Med Chem. 2018 Feb 8; 61(3): 1182–1203. Published online 2018 Jan 5. doi: 10.1021/acs.jmedchem.7b01654

PMCID:: PMC5965259

Abstract Article PDF–932K

Select item 84121425.

Lead Optimization of 3,5-Disubstituted-7-Azaindoles for the Treatment of Human African Trypanosomiasis

Dana M. Klug, Eftychia M. Mavrogiannaki, Katherine C. Forbes, Lisseth Silva, Rosario Diaz-Gonzalez, Guiomar Pérez-Moreno, Gloria Ceballos-Pérez, Raquel Garcia-Hernández, Cristina Bosch-Navarrete, Carlos Cordón-Obras, Claudia Gómez-Liñán, Andreu Saura, Jeremiah D. Momper, Maria Santos Martinez-Martinez, Pilar Manzano, Ali Syed, Nelly El-Sakkary, Conor R. Caffrey, Francisco Gamarro, Luis Miguel Ruiz-Perez, Dolores Gonzalez Pacanowska, Lori Ferrins, Miguel Navarro, Michael P. Pollastri

J Med Chem. Author manuscript; available in PMC 2022 Jul 8.

Published in final edited form as: J Med Chem. 2021 Jul 8; 64(13): 9404–9430. Published online 2021 Jun 22. doi: 10.1021/acs.jmedchem.1c00674

PMCID:: PMC8412142

Abstract Article PDF–1.3M

Select item 79185386.

Synthesis, Characterization, and Biological Evaluation of New Derivatives Targeting MbtI as Antitubercular Agents

Matteo Mori, Giovanni Stelitano, Laurent R. Chiarelli, Giulia Cazzaniga, Arianna Gelain, Daniela Barlocco, Elena Pini, Fiorella Meneghetti, Stefania Villa

Pharmaceuticals (Basel) 2021 Feb; 14(2): 155. Published online 2021 Feb 13. doi: 10.3390/ph14020155

PMCID:: PMC7918538

Abstract Article PDF–2.9M

Select item 97892097.

Design and optimization of 1H-1,2,3-triazole-4-carboxamides as novel, potent, and selective inverse agonists and antagonists of PXR

Yongtao Li, Wenwei Lin, Sergio C. Chai, Jing Wu, Kavya Annu, Taosheng Chen

J Med Chem. Author manuscript; available in PMC 2023 Dec 22.

Published in final edited form as: J Med Chem. 2022 Dec 22; 65(24): 16829–16859. Published online 2022 Dec 8. doi: 10.1021/acs.jmedchem.2c01640

PMCID:: PMC9789209

Abstract Article PDF–2.8M

Select item 105007048.

Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Lijun Song, Romain Merceron, Fabian Hulpia, Ainhoa Lucía, Begoña Gracia, Yanlin Jian, Martijn D.P. Risseeuw, Toon Verstraelen, Paul Cos, José A. Aínsa, Helena I. Boshoff, Hélène Munier-Lehmann, Savvas N. Savvides, Serge Van Calenbergh

Eur J Med Chem. Author manuscript; available in PMC 2023 Sep 14.

Published in final edited form as: Eur J Med Chem. 2021 Dec 5; 225: 113784. Published online 2021 Aug 18. doi: 10.1016/j.ejmech.2021.113784

PMCID:: PMC10500704

Abstract Article PDF–4.0M

Select item 44039329.

9H-Purine Scaffold Reveals Induced-Fit Pocket Plasticity of the BRD9 Bromodomain

Sarah Picaud, Maria Strocchia, Stefania Terracciano, Gianluigi Lauro, Jacqui Mendez, Danette L. Daniels, Raffaele Riccio, Giuseppe Bifulco, Ines Bruno, Panagis Filippakopoulos

J Med Chem. 2015 Mar 26; 58(6): 2718–2736. Published online 2015 Feb 22. doi: 10.1021/jm501893k

PMCID:: PMC4403932

Abstract Article PDF–4.8M

Select item 1150999810.

Pd-, Cu-, and Ni-Catalyzed Reactions: A Comprehensive Review of the Efficient Approaches towards the Synthesis of Antibacterial Molecules

Almeera Zia, Shehla Khalid, Nasir Rasool, Nayab Mohsin, Muhammad Imran, Sebastian Ionut Toma, Catalin Misarca, Oana Andreescu

Pharmaceuticals (Basel) 2024 Oct; 17(10): 1370. Published online 2024 Oct 15. doi: 10.3390/ph17101370

PMCID:: PMC11509998

Abstract Article PDF–23M

Select item 490193811.

A convenient route to symmetrically and unsymmetrically substituted 3,5-diaryl-2,4,6-trimethylpyridines via Suzuki–Miyaura cross-coupling reaction

Dariusz Błachut, Joanna Szawkało, Zbigniew Czarnocki

Beilstein J Org Chem. 2016; 12: 835–845. Published online 2016 Apr 28. doi: 10.3762/bjoc.12.82

PMCID:: PMC4901938

Abstract Article PDF–466K

Select item 831442312.

Discovery and Structure-Based Optimization of Benzimidazole-Derived Activators of SOS1-Mediated Nucleotide Exchange on RAS

Timothy R. Hodges, Jason R. Abbott, Andrew J. Little, Dhruba Sarkar, James M. Salovich, Jennifer E. Howes, Denis T. Akan, Jiqing Sai, Allison L. Arnold, Carrie Browning, Michael C. Burns, Tammy Sobolik, Qi Sun, Yugandhar Beesetty, Jesse A. Coker, Dirk Scharn, Heinz Stadtmueller, Olivia W. Rossanese, Jason Phan, Alex G. Waterson, Darryl B. McConnell, Stephen W. Fesik

J Med Chem. Author manuscript; available in PMC 2021 Jul 27.

Published in final edited form as: J Med Chem. 2018 Oct 11; 61(19): 8875–8894. Published online 2018 Sep 28. doi: 10.1021/acs.jmedchem.8b01108

PMCID:: PMC8314423

Abstract Article PDF–2.5M

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3-Bromo-5- AND (trifluoromethyl) AND phenylboronic acid (12)
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Piper psbJ-petA intergenic spacer region, partial sequence; chloroplast.
Piper psbJ-petA intergenic spacer region, partial sequence; chloroplast.
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