2,1-Benzisoxazole-7-carboxaldehyde - PMC

Select item 36971021.

Benzofuran-, benzothiophene-, indazole- and benzisoxazole- quinones: excellent substrates for NAD(P)H:quinone oxidoreductase 1

Jeffery J. Newsome, Mary Hassani, Elizabeth Swann, Jane M. Bibby, Howard D. Beall, Christopher J. Moody

Bioorg Med Chem. Author manuscript; available in PMC 2014 Jun 1.

Published in final edited form as: Bioorg Med Chem. 2013 Jun 1; 21(11): 2999–3009. Published online 2013 Apr 6. doi: 10.1016/j.bmc.2013.03.071

PMCID:: PMC3697102

Abstract Article PDF–2.8M

Select item 92339352.

Spiropyrimidinetrione DNA gyrase inhibitors with potent and selective antituberculosis activity

Preshendren Govender, Rudolf Müller, Kawaljit Singh, Virsinha Reddy, Charles J. Eyermann, Stephen Fienberg, Sandeep R. Ghorpade, Lizbé Koekemoer, Alissa Myrick, Dirk Schnappinger, Curtis Engelhart, Jaclynn Meshanni, Jo Ann W. Byl, Neil Osheroff, Vinayak Singh, Kelly Chibale, Gregory S. Basarab

J Med Chem. Author manuscript; available in PMC 2022 Jun 26.

Published in final edited form as: J Med Chem. 2022 May 12; 65(9): 6903–6925. Published online 2022 May 2. doi: 10.1021/acs.jmedchem.2c00266

PMCID:: PMC9233935

Abstract Article PDF–2.7M

Select item 27716983.

Structurally Simple Inhibitors of Lanosterol 14α-Demethylase Are Efficacious In a Rodent Model of Acute Chagas Disease

Praveen Kumar Suryadevara, Srinivas Olepu, Jeffrey W. Lockman, Junko Ohkanda, Mandana Karimi, Christophe L. M. J. Verlinde, James M. Kraus, Jan Schoepe, Wesley C. Van Voorhis, Andrew D. Hamilton, Frederick S. Buckner, Michael H. Gelb

J Med Chem. Author manuscript; available in PMC 2009 Nov 2.

Published in final edited form as: J Med Chem. 2009 Jun 25; 52(12): 3703–3715. doi: 10.1021/jm900030h

PMCID:: PMC2771698

Abstract Article PDF–2.2M

Select item 100755064.

Synthesis and biological evaluation of flavonoid-based IP6K2 inhibitors

Myunghwan Ahn, Seung Eun Park, Jiyeon Choi, Jiahn Choi, Doyoung Choi, Dongju An, Hayoung Jeon, Soowhan Oh, Kiho Lee, Jaehoon Kim, Jaebong Jang, Seyun Kim, Youngjoo Byun

J Enzyme Inhib Med Chem. 2023; 38(1): 2193866. Published online 2023 Apr 4. doi: 10.1080/14756366.2023.2193866