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Wee1 Inhibitor response

MedGen UID:
1001571
Concept ID:
CN322757
Sign or Symptom
Drug:
Wee1 Inhibitor
MedGen UID:
981754
Concept ID:
CN298257
Pharmacologic Substance

Professional guidelines

PubMed

Chao Y, Chen Y, Zheng W, Demanelis K, Liu Y, Connelly JA, Wang H, Li S, Wang QJ
Oncogene 2024 Mar;43(11):789-803. Epub 2024 Jan 25 doi: 10.1038/s41388-024-02939-z. PMID: 38273024
Chien W, Tyner JW, Gery S, Zheng Y, Li LY, Gopinatha Pillai MS, Nam C, Bhowmick NA, Lin DC, Koeffler HP
J Ovarian Res 2023 Apr 22;16(1):80. doi: 10.1186/s13048-023-01160-y. PMID: 37087441Free PMC Article
van Harten AM, de Boer DV, Martens-de Kemp SR, Buijze M, Ganzevles SH, Hunter KD, Leemans CR, van Beusechem VW, Wolthuis RMF, de Menezes RX, Brakenhoff RH
Sci Rep 2020 Feb 11;10(1):2330. doi: 10.1038/s41598-020-58509-2. PMID: 32047167Free PMC Article

Recent clinical studies

Etiology

Pearson ADJ, Federico S, Gatz SA, Ortiz M, Lesa G, Scobie N, Gounaris I, Weiner SL, Weigel B, Unger TJ, Stewart E, Smith M, Slotkin EK, Reaman G, Pappo A, Nysom K, Norga K, McDonough J, Marshall LV, Ludwinski D, Ligas F, Karres D, Kool M, Horner TJ, Henssen A, Heenen D, Hawkins DS, Gore L, Bender JG, Galluzzo S, Fox E, de Rojas T, Davies BR, Chakrabarti J, Carmichael J, Bradford D, Blanc P, Bernardi R, Benchetrit S, Akindele K, Vassal G
Eur J Cancer 2023 Sep;190:112950. Epub 2023 Jun 21 doi: 10.1016/j.ejca.2023.112950. PMID: 37441939
Bauer TM, Moore KN, Rader JS, Simpkins F, Mita AC, Beck JT, Hart L, Chu Q, Oza A, Tinker AV, Imedio ER, Kumar S, Mugundu G, Jenkins S, Chmielecki J, Jones S, Spigel D, Fu S
Target Oncol 2023 Jul;18(4):517-530. Epub 2023 Jun 6 doi: 10.1007/s11523-023-00965-7. PMID: 37278879Free PMC Article
Schutte T, Embaby A, Steeghs N, van der Mierden S, van Driel W, Rijlaarsdam M, Huitema A, Opdam F
Cancer Treat Rev 2023 Apr;115:102531. Epub 2023 Mar 3 doi: 10.1016/j.ctrv.2023.102531. PMID: 36893690
Fu S, Yao S, Yuan Y, Previs RA, Elias AD, Carvajal RD, George TJ, Yuan Y, Yu L, Westin SN, Xing Y, Dumbrava EE, Karp DD, Piha-Paul SA, Tsimberidou AM, Ahnert JR, Takebe N, Lu K, Keyomarsi K, Meric-Bernstam F
J Clin Oncol 2023 Mar 20;41(9):1725-1734. Epub 2022 Dec 5 doi: 10.1200/JCO.22.00830. PMID: 36469840Free PMC Article
Lindemann A, Takahashi H, Patel AA, Osman AA, Myers JN
J Dent Res 2018 Jun;97(6):635-644. Epub 2018 Feb 28 doi: 10.1177/0022034518759068. PMID: 29489434Free PMC Article

Diagnosis

Li J, Lu J, Xu M, Yang S, Yu T, Zheng C, Huang X, Pan Y, Chen Y, Long J, Zhang C, Huang H, Dai Q, Li B, Wang W, Yao S, Pan C
J Clin Invest 2023 Jan 17;133(2) doi: 10.1172/JCI161544. PMID: 36378528Free PMC Article
Durinikova E, Reilly NM, Buzo K, Mariella E, Chilà R, Lorenzato A, Dias JML, Grasso G, Pisati F, Lamba S, Corti G, Degasperi A, Cancelliere C, Mauri G, Andrei P, Linnebacher M, Marsoni S, Siena S, Sartore-Bianchi A, Nik-Zainal S, Di Nicolantonio F, Bardelli A, Arena S
Clin Cancer Res 2022 Sep 1;28(17):3874-3889. doi: 10.1158/1078-0432.CCR-22-0875. PMID: 35881546Free PMC Article
Guo E, Xiao R, Wu Y, Lu F, Liu C, Yang B, Li X, Fu Y, Wang Z, Li Y, Huang Y, Li F, Wu X, You L, Qin T, Lu Y, Huang X, Ma D, Mills GB, Sun C, Chen G
J Exp Med 2022 Jan 3;219(1) Epub 2021 Nov 26 doi: 10.1084/jem.20210789. PMID: 34825915Free PMC Article
Cleary JM, Aguirre AJ, Shapiro GI, D'Andrea AD
Mol Cell 2020 Jun 18;78(6):1070-1085. Epub 2020 May 26 doi: 10.1016/j.molcel.2020.04.035. PMID: 32459988Free PMC Article
Pilié PG, Tang C, Mills GB, Yap TA
Nat Rev Clin Oncol 2019 Feb;16(2):81-104. doi: 10.1038/s41571-018-0114-z. PMID: 30356138Free PMC Article

Therapy

da Costa AABA, Chowdhury D, Shapiro GI, D'Andrea AD, Konstantinopoulos PA
Nat Rev Drug Discov 2023 Jan;22(1):38-58. Epub 2022 Oct 6 doi: 10.1038/s41573-022-00558-5. PMID: 36202931
Cheng B, Pan W, Xing Y, Xiao Y, Chen J, Xu Z
Eur J Med Chem 2022 Feb 15;230:114109. Epub 2022 Jan 12 doi: 10.1016/j.ejmech.2022.114109. PMID: 35051747
Smith HL, Southgate H, Tweddle DA, Curtin NJ
Expert Rev Mol Med 2020 Jun 8;22:e2. doi: 10.1017/erm.2020.3. PMID: 32508294
Cleary JM, Aguirre AJ, Shapiro GI, D'Andrea AD
Mol Cell 2020 Jun 18;78(6):1070-1085. Epub 2020 May 26 doi: 10.1016/j.molcel.2020.04.035. PMID: 32459988Free PMC Article
Pilié PG, Tang C, Mills GB, Yap TA
Nat Rev Clin Oncol 2019 Feb;16(2):81-104. doi: 10.1038/s41571-018-0114-z. PMID: 30356138Free PMC Article

Prognosis

Schutte T, Embaby A, Steeghs N, van der Mierden S, van Driel W, Rijlaarsdam M, Huitema A, Opdam F
Cancer Treat Rev 2023 Apr;115:102531. Epub 2023 Mar 3 doi: 10.1016/j.ctrv.2023.102531. PMID: 36893690
Li J, Lu J, Xu M, Yang S, Yu T, Zheng C, Huang X, Pan Y, Chen Y, Long J, Zhang C, Huang H, Dai Q, Li B, Wang W, Yao S, Pan C
J Clin Invest 2023 Jan 17;133(2) doi: 10.1172/JCI161544. PMID: 36378528Free PMC Article
Xu H, George E, Kinose Y, Kim H, Shah JB, Peake JD, Ferman B, Medvedev S, Murtha T, Barger CJ, Devins KM, D'Andrea K, Wubbenhorst B, Schwartz LE, Hwang WT, Mills GB, Nathanson KL, Karpf AR, Drapkin R, Brown EJ, Simpkins F
Cell Rep Med 2021 Sep 21;2(9):100394. Epub 2021 Sep 23 doi: 10.1016/j.xcrm.2021.100394. PMID: 34622231Free PMC Article
Cleary JM, Aguirre AJ, Shapiro GI, D'Andrea AD
Mol Cell 2020 Jun 18;78(6):1070-1085. Epub 2020 May 26 doi: 10.1016/j.molcel.2020.04.035. PMID: 32459988Free PMC Article
Pilié PG, Tang C, Mills GB, Yap TA
Nat Rev Clin Oncol 2019 Feb;16(2):81-104. doi: 10.1038/s41571-018-0114-z. PMID: 30356138Free PMC Article

Clinical prediction guides

Li J, Lu J, Xu M, Yang S, Yu T, Zheng C, Huang X, Pan Y, Chen Y, Long J, Zhang C, Huang H, Dai Q, Li B, Wang W, Yao S, Pan C
J Clin Invest 2023 Jan 17;133(2) doi: 10.1172/JCI161544. PMID: 36378528Free PMC Article
Durinikova E, Reilly NM, Buzo K, Mariella E, Chilà R, Lorenzato A, Dias JML, Grasso G, Pisati F, Lamba S, Corti G, Degasperi A, Cancelliere C, Mauri G, Andrei P, Linnebacher M, Marsoni S, Siena S, Sartore-Bianchi A, Nik-Zainal S, Di Nicolantonio F, Bardelli A, Arena S
Clin Cancer Res 2022 Sep 1;28(17):3874-3889. doi: 10.1158/1078-0432.CCR-22-0875. PMID: 35881546Free PMC Article
Xu H, George E, Kinose Y, Kim H, Shah JB, Peake JD, Ferman B, Medvedev S, Murtha T, Barger CJ, Devins KM, D'Andrea K, Wubbenhorst B, Schwartz LE, Hwang WT, Mills GB, Nathanson KL, Karpf AR, Drapkin R, Brown EJ, Simpkins F
Cell Rep Med 2021 Sep 21;2(9):100394. Epub 2021 Sep 23 doi: 10.1016/j.xcrm.2021.100394. PMID: 34622231Free PMC Article
Cleary JM, Aguirre AJ, Shapiro GI, D'Andrea AD
Mol Cell 2020 Jun 18;78(6):1070-1085. Epub 2020 May 26 doi: 10.1016/j.molcel.2020.04.035. PMID: 32459988Free PMC Article
Pilié PG, Tang C, Mills GB, Yap TA
Nat Rev Clin Oncol 2019 Feb;16(2):81-104. doi: 10.1038/s41571-018-0114-z. PMID: 30356138Free PMC Article

Recent systematic reviews

Wang Z, Li W, Li F, Xiao R
J Cancer Res Clin Oncol 2024 Jan 17;150(1):13. doi: 10.1007/s00432-023-05527-y. PMID: 38231277Free PMC Article
Schutte T, Embaby A, Steeghs N, van der Mierden S, van Driel W, Rijlaarsdam M, Huitema A, Opdam F
Cancer Treat Rev 2023 Apr;115:102531. Epub 2023 Mar 3 doi: 10.1016/j.ctrv.2023.102531. PMID: 36893690

Supplemental Content

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    Clinical resources

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