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Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.

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Probe Reports from the NIH Molecular Libraries Program [Internet].

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Table 6Receptor Paneling of KOP agonist Probes 1 [ML139] CID5236771 & 2 [ML138] CID44601470 through the PDSP (Bryan Roth, PI)

ReceptorProbe Ki (nM)
ML139ML138
5ht1a
5ht1b
5ht1d
5ht1e
5ht2a
5ht2b1,237
5ht2c
5ht3
5ht5a4,986
5ht6
5ht7
Alpha1A
Alpha1B
Alpha1D
Alpha2A5,525
Alpha2B9,601
Alpha2C
Beta1
Beta2
Beta37,312
BZP Rat Brain Site
D11,796
D2
D3
D4
D57018
DAT
DOR1,315484.1
H1
H2
H3
H4
KOR0.790.23
M1
M2
M3
M4
M5
MOR671.1773.3
NET
SERT
Sigma 1

Image ml139fu20.jpg Green: Ki > 10,000 or 1ary screen missed

Image ml139fu21.jpg Orange: 2ndary assay pending

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