Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane assessed as inhibition constant
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane assessed as inhibition constant measured for 150 mins
Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane assessed as inhibition constant measured after 120 mins by scintillation counting method
Assay data:5 Active, 2 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane assessed as inhibition constant measured for 150 mins in presence of haloperidol
Assay data:10 Active, 1 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
Antagonist activity at histamine H1 receptor in guinea pig isolated trachea assessed as change in histamine-induced contraction
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Effect on fingolimod-induced shortening of AERP in guinea pig model assessed as restoration of shortened AERP measured at 30 to 60 mins
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane assessed as inhibition constant incubated for 120 mins
Assay data:11 Active, 11 Activity ≤ 1 µM, 12 Tested
Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes assessed as inhibition constant by Wallac 1450 MicroBeta liquid scintillation counter
Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes assessed as inhibition constant by competitive binding assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of transglutaminase in guinea pig liver assessed as inhibition constant using Z-Gln-Gly as substrate by Michaelis-Menten analysis
Assay data:2 Tested
SummaryPubMed Citation
Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membranes measured after 120 mins by scintillation counting method
Assay data:9 Active, 7 Activity ≤ 1 µM, 9 Tested
Displacement of [3H]pentazocine from guinea pig brain membrane sigma 1 receptor incubated for 150 mins
Displacement of [3H]pentazocine from guinea pig brain membrane sigma 1 receptor incubated for 120 mins
Transporter, Adenosine Eurofins Panlabs panel
Summary
Serotonin (5-Hydroxytryptamine) 5-HT4 Eurofins Panlabs panel
SummaryRelated BioAssays by Target
Leukotriene LTC4 Synthase Eurofins Panlabs panel
Displacement of [3H]pentazocine from sigma 1 receptor expressed in guinea pig brain membranes assessed as inhibition constant incubated for 150 mins by radioligand binding assay
Displacement of [3H]pentazocine from sigma 1 receptor expressed in guinea pig brain membranes assessed as inhibition constant by radioligand binding assay
Assay data:11 Active, 3 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested
Binding affinity to sigma 1 receptor expressed in guinea pig brain
Assay data:4 Active, 1 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 4 Tested
Inhibition of superoxide anion radical release in guinea pig peritoneal macrophages
Assay data:11 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on