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Agonist activity at human beta2 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulation
Assay data:39 Active, 39 Activity ≤ 1 nM, 39 Activity ≤ 1 µM, 39 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at human beta2 adrenergic receptor expressed in HEK293 cells assessed as increase in cAMP accumulation after 60 mins by HTRF assay
Assay data:26 Active, 24 Activity ≤ 1 nM, 26 Activity ≤ 1 µM, 26 Tested
Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident proteome: Secreted ER Calcium Modulated Protein (SERCaMP) assay
Assay data:41 Active, 8 Activity ≤ 1 nM, 357 Activity ≤ 1 µM, 11292 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Depositor
Assay data:27 Active, 1 Activity ≤ 1 nM, 27 Activity ≤ 1 µM, 27 Tested
Agonist activity at human beta2-AR expressed in CHOK1 cells co-expressing Galpha15 measured after 21 secs to 120 secs by Calcium-4 dye based FLIPR assay
Assay data:3 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 3 Tested
Unbound Cmax in human plasma
Assay data:66 Active, 5 Activity ≤ 1 nM, 45 Activity ≤ 1 µM, 85 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Agonist activity at human beta2 adrenergic receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation
Assay data:12 Active, 2 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 13 Tested
Agonist activity at human recombinant adrenergic beta2 receptor expressed in CHO cells assessed as stimulation of cAMP level after 1 hr by enzyme immunoassay
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 13 Tested
Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as cAMP accumulation
Assay data:17 Active, 1 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 22 Tested
Agonist activity at human cloned adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulation
Assay data:22 Active, 1 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 22 Tested
Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation
Assay data:25 Active, 1 Activity ≤ 1 nM, 49 Activity ≤ 1 µM, 51 Tested
Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation
Assay data:49 Active, 10 Activity ≤ 1 nM, 51 Activity ≤ 1 µM, 51 Tested
Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassay
Assay data:45 Active, 38 Activity ≤ 1 nM, 45 Activity ≤ 1 µM, 45 Tested
Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassay
Assay data:28 Active, 1 Activity ≤ 1 nM, 45 Activity ≤ 1 µM, 45 Tested
Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assay
Assay data:52 Active, 38 Activity ≤ 1 nM, 52 Activity ≤ 1 µM, 52 Tested
Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assay
Assay data:42 Active, 1 Activity ≤ 1 nM, 50 Activity ≤ 1 µM, 50 Tested
Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIA
Assay data:28 Active, 1 Activity ≤ 1 nM, 42 Activity ≤ 1 µM, 43 Tested
Agonist activity at human beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIA
Assay data:42 Active, 11 Activity ≤ 1 nM, 43 Activity ≤ 1 µM, 43 Tested
Activity at human beta-1 adrenergic receptor expressed in CHO cells by stimulation of cAMP production
Assay data:15 Active, 1 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 15 Tested
Activity at human beta-2 adrenergic receptor expressed in CHO cells by stimulation of cAMP production
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