BioAssays, Active for PubChem Compound (Select 782728) - PubChem BioAssay - NCBI

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Items: 6

Select item 14671501.

Displacement of (+)-[3H]-ditolylguanidine from recombinant rat sigma 2 receptor expressed in rat PC12 cell membranes after 90 mins in presence of sigma 1 receptor blocker (+)-SKF-10047 by scintillation counting method

Source:: ChEMBL

Protein Target:: Sigma intracellular receptor 2

Assay data:7 Active, 6 Activity ≤ 1 µM, 7 Tested

AID:: 1467150

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14671492.

Displacement of (+)-[3H]-pentazocine from recombinant human sigma 1 receptor expressed in baculovirus infected Sf9 insect cell membranes after 90 mins by scintillation counting method

Source:: ChEMBL

Protein Target:: Sigma non-opioid intracellular receptor 1

Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested

AID:: 1467149

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 6241263.

Fluorescence-based cell-based primary high throughput screening assay to identify positive allosteric modulators (PAMs) of the human cholinergic receptor, muscarinic 4 (CHRM4)

Source:: The Scripps Research Institute Molecular Screening Center

Protein Target:: muscarinic acetylcholine receptor M4

Assay data:1450 Active, 364131 Tested

AID:: 624126

Summary Compounds, Active PubMed Citation Related BioAssays by Depositor Related BioAssays by Same Project Related BioAssays by Target

Select item 5043394.

qHTS Assay for Inhibitors of JMJD2A-Tudor Domain

Source:: National Center for Advancing Translational Sciences (NCATS)

Protein Target:: Chain A, JmjC domain-containing histone demethylation protein 3A

Assay data:17028 Active, 1 Activity ≤ 1 nM, 596 Activity ≤ 1 µM, 388413 Tested

AID:: 504339

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Depositor Related BioAssays by Same Project Related BioAssays by Target

Select item 5043325.

qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a

Source:: National Center for Advancing Translational Sciences (NCATS)

Protein Target:: euchromatic histone-lysine N-methyltransferase 2

Assay data:31109 Active, 1 Activity ≤ 1 nM, 5166 Activity ≤ 1 µM, 353740 Tested

AID:: 504332

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Depositor Related BioAssays by Same Project Related BioAssays by Target

Select item 19966.

Aqueous Solubility from MLSMR Stock Solutions

Source:: Burnham Center for Chemical Genomics

Assay data:40286 Active, 57859 Tested

AID:: 1996

Summary Compounds, Active PubMed Citation

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Target

Proteins (3)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (6)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (4)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (4)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (1)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (3)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (2)
BioAssays extracted from the literature
NIH MLP (4)
BioAssays deposited by the NIH Molecular Libraries Program

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BioAssays, Active for PubChem Compound (Select 782728) (6)
PubChem BioAssay
Protein Links for OMIM (Select 246900) (0)
Protein
Book Links for OMIM (Select 246900) (3)
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Rattus norvegicus MAS-related GPR, member F (Mrgprf), mRNA
Rattus norvegicus MAS-related GPR, member F (Mrgprf), mRNA
gi|24308469|ref|NM_153722.1|

Nucleotide

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