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Trypanocidal activity against Trypanosoma cruzi MHOM/MX/1994/Ninoa assessed as inhibition of parasite growth measured after 48 hrs by MTT assay
Assay data:4 Active, 10 Tested
SummaryCompounds, ActivePubMed Citation
P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen
Assay data:1430 Active, 11 Activity ≤ 1 nM, 385 Activity ≤ 1 µM, 10968 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
Drug repurposing screens with cells derived from glioblastoma tumor samples
Assay data:1237 Active, 3 Activity ≤ 1 nM, 360 Activity ≤ 1 µM, 3733 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary
Assay data:589 Active, 16 Activity ≤ 1 nM, 99 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway: Summary
Assay data:670 Active, 220 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary
Assay data:372 Active, 6 Activity ≤ 1 nM, 228 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line
Assay data:1084 Active, 8 Activity ≤ 1 nM, 330 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway
Assay data:589 Active, 14 Activity ≤ 1 nM, 591 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line
Assay data:461 Active, 11 Activity ≤ 1 nM, 217 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway
Assay data:233 Active, 2 Activity ≤ 1 nM, 236 Activity ≤ 1 µM, 10486 Tested
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line
Assay data:2501 Active, 1 Activity ≤ 1 nM, 348 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway: Summary
Assay data:460 Active, 10486 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule antagonists of the glucocorticoid receptor (GR) signaling pathway
Assay data:406 Active, 2 Activity ≤ 1 nM, 281 Activity ≤ 1 µM, 10486 Tested
Displacement of [3H]5alpha dihydrotestosterone from human sex hormone binding globulin
Assay data:87 Active, 17 Activity ≤ 1 nM, 79 Activity ≤ 1 µM, 90 Tested
Binding affinity at AR
Assay data:17 Active, 13 Activity ≤ 1 µM, 17 Tested
Agonist activity at ERbeta expressed in HEK293 cells by transactivation assay
Assay data:15 Active, 17 Activity ≤ 1 µM, 17 Tested
Agonist activity at ERalpha expressed in HEK293 cells by transactivation assay
Assay data:8 Active, 1 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 17 Tested
Binding affinity at human recombinant ERbeta
Assay data:17 Active, 15 Activity ≤ 1 µM, 18 Tested
Binding affinity at human recombinant ERalpha
Assay data:13 Active, 5 Activity ≤ 1 µM, 17 Tested
Inhibitory activity against AR
Assay data:24 Active, 15 Activity ≤ 1 µM, 27 Tested
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