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Selectivity index, ratio IC50 for recombinant human MAO-B to IC50 for recombinant human MAO-A
Assay data:14 Tested
SummaryPubMed Citation
Inhibition of recombinant human MAO-B expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by fluorescence spectrophotometric assay
Assay data:6 Active, 14 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of recombinant human MAO-A expressed in baculovirus infected BTI insect cells using kynuramine as substrate after 20 mins by fluorescence spectrophotometric assay
Assay data:11 Active, 3 Activity ≤ 1 µM, 26 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antiproliferative activity against human A-431 cells overexpressing EGFR assessed as reduction in cell survival at 10 uM
Inhibition of His-tagged HSD17B13 (unknown origin) using LTB3 as substrate incubated for 1 hr and measured after 1 hr by fluorescence based assay
Assay data:3 Active, 4 Tested
SummaryCompounds, Active
Inhibition of His-tagged HSD17B13 (unknown origin) using estradiol as substrate incubated for 2 hrs and measured by LC-MS/MS analysis
Assay data:3 Active, 1 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Ratio of Ki for inhibition of His-tagged HSD17B13 (unknown origin) using LTB3 as substrate to Ki for His-tagged HSD17B13 (unknown origin) using estradiol as substrate
Assay data:4 Tested
Summary
Cell-based high-throughput assay to identify small molecules that inhibit phospholipid biosynthesis in animal cells 2: screen of the Analyticon library.
Assay data:3 Active, 495 Tested
SummaryCompounds, ActiveRelated BioAssays by Depositor
Primary cell-based high-throughput screening assay for identification of small molecule agonists of Aedes aegypti NPYLR7 [Small Molecule Inhibitors of Mosquito Biting Behavior]
Assay data:412 Active, 270665 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Depositor
CCRIS mutagenicity studies
Assay data:4929 Active, 8266 Tested
human cGAS chemiluminescence screen
Assay data:234 Active, 287414 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
mouse cGAS RapidFire screen
Assay data:231 Active, 125931 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition of human recombinant UGT1A1 expressed in HEK293 cells assessed as reduction in estradiol 3-glucuronidation by LC-MS/MS method
Assay data:4 Active, 16 Tested
Inhibition of human recombinant UGT1A1 expressed in HEK293 cells assessed as reduction in bilirubin glucuronidation by LC-MS/MS method
Assay data:5 Active, 16 Tested
Specific activity of expressed human recombinant UGT2B15
Assay data:111 Tested
SummaryPubMed CitationRelated BioAssays by Target
Specific activity of expressed human recombinant UGT2A1
Assay data:42 Tested
Specific activity of expressed human recombinant UGT1A10
Assay data:117 Tested
Specific activity of expressed human recombinant UGT1A9
Assay data:122 Tested
Specific activity of expressed human recombinant UGT1A8
Specific activity of expressed human recombinant UGT1A6
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