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Inhibition of His6-tagged recombinant human GALK expressed in Escherichia coli HMS174 (DE3) at 5 to 15 uM incubated for 60 mins using galactose and ATP by Kinase-Glo reagent based assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Agonist activity at human N-terminal HA-tagged P2Y2 receptor expressed in 1321N1 cells
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB
Assay data:3916 Active, 206 Activity ≤ 1 nM, 1830 Activity ≤ 1 µM, 3916 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Antioxidant activity assessed as inhibiton of Fe2+-induced Fenton reaction-mediated hydroxyl radical formation from H2O2 relative to ATP
Assay data:1 Tested
SummaryPubMed Citation
Antioxidant activity assessed as inhibiton of Fe2+-induced Fenton reaction-mediated hydroxyl radical formation from H2O2 relative to trolox
Agonist activity at P2Y11 receptor expressed in 1321N1 cells assessed as cytosolic calcium level
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )
Assay data:11 Active, 6 Activity ≤ 1 µM, 11 Tested
Antagonist activity against phospholipase C coupled rat P2Y purinoceptor 12 (P2Y12)
Assay data:7 Active, 4 Activity ≤ 1 µM, 12 Tested
Agonist activity against phospholipase C coupled human P2Y purinoceptor 11 (P2Y11)
Assay data:4 Active, 10 Tested
Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of turkey erythrocytes
Assay data:14 Active, 1 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 17 Tested
Evaluated for agonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 2 (P2Y2)
Assay data:4 Active, 3 Activity ≤ 1 µM, 12 Tested
Antagonist activity against recombinant rat P2X purinoceptor 6 (P2X6 )
Assay data:3 Active, 2 Activity ≤ 1 µM, 7 Tested
Antagonist activity against recombinant rat P2X purinoceptor 5 (P2X5)
Assay data:5 Active, 3 Activity ≤ 1 µM, 7 Tested
Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 30 uM, expressed in Xenopus oocytes
Assay data:3 Active, 1 Activity ≤ 1 µM, 5 Tested
Antagonist activity against recombinant human P2X purinoceptor 3 (P2X3 )
Assay data:9 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 11 Tested
Antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 10 uM, expressed in Xenopus oocytes
Assay data:4 Active, 1 Activity ≤ 1 µM, 7 Tested
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