BioAssays for PubChem Compound (Select 3779) - PubChem BioAssay - NCBI

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Select item 19618781.

Binding affinity towards human HRH3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Histamine H3 receptor

Assay data:41 Active, 7 Activity ≤ 1 µM, 993 Tested

AID:: 1961878

Summary Related BioAssays by Target

Select item 19618682.

Binding affinity towards human ADRA1A in an in vitro assay with cellular components (NIBR assay) measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Alpha-1A adrenergic receptor

Assay data:49 Active, 29 Activity ≤ 1 µM, 231 Tested

AID:: 1961868

Summary Related BioAssays by Target

Select item 19618603.

Binding affinity towards human AGTR1 in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Type-1 angiotensin II receptor

Assay data:3 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 20 Tested

AID:: 1961860

Summary Related BioAssays by Target

Select item 19618594.

Binding affinity towards human DRD1 in an in vitro assay with cellular components (NIBR assay) measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(1A) dopamine receptor

Assay data:35 Active, 19 Activity ≤ 1 µM, 305 Tested

AID:: 1961859

Summary Related BioAssays by Target

Select item 19618575.

Binding affinity towards human CHRM2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Muscarinic acetylcholine receptor M2

Assay data:58 Active, 2 Activity ≤ 1 nM, 37 Activity ≤ 1 µM, 301 Tested

AID:: 1961857

Summary Related BioAssays by Target

Select item 19618566.

Binding affinity towards human DRD3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: D(3) dopamine receptor

Assay data:176 Active, 1 Activity ≤ 1 nM, 87 Activity ≤ 1 µM, 1215 Tested

AID:: 1961856

Summary Related BioAssays by Target

Select item 19618557.

Compound was evaluated for inhibition of human PDE3A in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: cGMP-inhibited 3',5'-cyclic phosphodiesterase A

Assay data:49 Active, 5 Activity ≤ 1 µM, 1243 Tested

AID:: 1961855

Summary Related BioAssays by Target

Select item 19618538.

Binding affinity towards human HTR1A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1A

Assay data:56 Active, 33 Activity ≤ 1 µM, 377 Tested

AID:: 1961853

Summary Related BioAssays by Target

Select item 19618529.

Compound was evaluated for inhibition of human MAOA in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Amine oxidase [flavin-containing] A

Assay data:28 Active, 4 Activity ≤ 1 µM, 1218 Tested

AID:: 1961852

Summary Related BioAssays by Target

Select item 196185110.

Binding affinity towards human OPRM1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Mu-type opioid receptor

Assay data:60 Active, 9 Activity ≤ 1 µM, 766 Tested

AID:: 1961851

Summary Related BioAssays by Target

Select item 196185011.

Binding affinity towards human ADRA2A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Alpha-2A adrenergic receptor

Assay data:63 Active, 20 Activity ≤ 1 µM, 323 Tested

AID:: 1961850

Summary Related BioAssays by Target

Select item 196184912.

Binding affinity towards human SLC6A4 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:148 Active, 75 Activity ≤ 1 µM, 1194 Tested

AID:: 1961849

Summary Related BioAssays by Target

Select item 196184813.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:123 Active, 40 Activity ≤ 1 µM, 1197 Tested

AID:: 1961848

Summary Related BioAssays by Target

Select item 196184714.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:119 Active, 21 Activity ≤ 1 µM, 1213 Tested

AID:: 1961847

Summary Related BioAssays by Target

Select item 196184615.

Binding affinity towards human TBXA2R in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:14 Active, 2 Activity ≤ 1 µM, 1022 Tested

AID:: 1961846

Summary Related BioAssays by Target

Select item 196184116.

Binding affinity towards human TACR1 in an in vitro assay with cellular components measured by membrane filtration

Source:: ChEMBL

Protein Target:: Substance-P receptor

Assay data:19 Active, 4 Activity ≤ 1 µM, 218 Tested

AID:: 1961841

Summary Related BioAssays by Target

Select item 196183717.

Binding affinity towards human SLC29A1 in an in vitro assay with cellular components measured by scintillation proximity assay

Source:: ChEMBL

Protein Target:: Equilibrative nucleoside transporter 1

Assay data:20 Active, 4 Activity ≤ 1 µM, 1115 Tested

AID:: 1961837

Summary Related BioAssays by Target

Select item 196182718.

Compound was evaluated for inhibition of human PTGS2 in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 2

Assay data:79 Active, 12 Activity ≤ 1 µM, 1183 Tested

AID:: 1961827

Summary Related BioAssays by Target

Select item 196182519.

Compound was evaluated for inhibition of rat Ptgs1 in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 1

Assay data:74 Active, 33 Activity ≤ 1 µM, 1201 Tested

AID:: 1961825

Summary Related BioAssays by Target

Select item 196181920.

Binding affinity towards human PGR in an in vitro cell free assay measured by fluorescence polarization method in vitro cell free assay

Source:: ChEMBL

Protein Target:: Progesterone receptor

Assay data:15 Active, 5 Activity ≤ 1 µM, 357 Tested

AID:: 1961819

Summary Related BioAssays by Target

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Target

Proteins (284)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (883)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (219)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (641)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Summary (63)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (807)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (84)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (296)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (505)
BioAssays extracted from the literature
NIH MLP (191)
BioAssays deposited by the NIH Molecular Libraries Program
Other (522)
BioAssays deposited by other experimentalists

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