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Summary
Human kisspeptin (KISS1R) small molecule agonists, calcium flux assay in KISS1R-HEK293 cells: Summary
Assay data:16 Active, 9667 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Same Project
Human gonadotropin-releasing hormone receptor (GnRHR) small molecule agonists, calcium flux assay in GnRHR-HEK293 cells: Summary
Assay data:109 Active, 9667 Tested
G protein-coupled receptor (GPCR) small molecule agonists, calcium flux assay: HEK293 wild type cell line counter screen
Assay data:47 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
Human kisspeptin (KISS1R) small molecule agonists, calcium flux assay in KISS1R-HEK293 cells
Assay data:55 Active, 2 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 9667 Tested
Human gonadotropin-releasing hormone receptor (GnRHR) small molecule agonists, calcium flux assay in GnRHR-HEK293 cells
Assay data:169 Active, 2 Activity ≤ 1 nM, 27 Activity ≤ 1 µM, 9667 Tested
High-throughput screening primary assay to identify small molecule activators of human guanylyl cyclase B (GC-B) receptor activity
Assay data:399 Active, 370620 Tested
SummaryCompounds, Active
Dual reporter qHTS for antagonist of Pregnane X Receptor (hPXR) against the NCATS DSHEA and TCM libraries: Fluorescence Readout
Assay data:28 Active, 4 Activity ≤ 1 µM, 964 Tested
SummaryPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Dual reporter qHTS for antagonist of Pregnane X Receptor (hPXR) against the NCATS DSHEA and TCM libraries: Luminescence Readout
Assay data:11 Active, 8 Activity ≤ 1 µM, 964 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Dual reporter qHTS for agonist of Pregnane X Receptor (hPXR) against the NCATS DSHEA and TCM libraries: Luminescence readout
Assay data:82 Active, 964 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Dual reporter qHTS for agonist of Pregnane X Receptor (hPXR) against the NCATS DSHEA and TCM libraries: Fluorescence readout
Assay data:1 Active, 3 Activity ≤ 1 µM, 964 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
qHTS Counterscreen for compound interference against the NCATS DSHEA and TCM libraries
Assay data:1 Active, 1 Activity ≤ 1 µM, 964 Tested
SummaryPubMed CitationRelated BioAssays by Depositor
KB-8-5-11 P-gp reporter qHTS against the NCATS DSHEA and TCM libraries
Assay data:27 Active, 1 Activity ≤ 1 µM, 964 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Depositor
qHTS for inhibitors of CYPIA2 against the NCATS DSHEA and TCM libraries
Assay data:275 Active, 13 Activity ≤ 1 µM, 964 Tested
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