BioAssays for PubChem Compound (Select 2993) - PubChem BioAssay - NCBI

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Select item 19618451.

Antagonist activity at human TBXA2R in an in vitro cell-based assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:34 Active, 15 Activity ≤ 1 µM, 906 Tested

AID:: 1961845

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618442.

Agonist activity at human TBXA2R in an in vitro cell-based assay (CRO assay) measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:13 Active, 8 Activity ≤ 1 µM, 927 Tested

AID:: 1961844

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618403.

Binding affinity towards human SLC6A4 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:99 Active, 36 Activity ≤ 1 µM, 927 Tested

AID:: 1961840

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618394.

Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:128 Active, 38 Activity ≤ 1 µM, 927 Tested

AID:: 1961839

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618385.

Binding affinity towards human SLC6A2 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:137 Active, 27 Activity ≤ 1 µM, 927 Tested

AID:: 1961838

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618286.

Compound was evaluated for inhibition of human PTGS1 in an in vitro cell free assay measured by fluorescence method

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 1

Assay data:80 Active, 33 Activity ≤ 1 µM, 924 Tested

AID:: 1961828

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618267.

Compound was evaluated for inhibition of human PTGS1 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: Prostaglandin G/H synthase 1

Assay data:96 Active, 35 Activity ≤ 1 µM, 927 Tested

AID:: 1961826

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618208.

Binding affinity towards human PGR in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Progesterone receptor

Assay data:87 Active, 51 Activity ≤ 1 µM, 927 Tested

AID:: 1961820

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19618149.

Compound was evaluated for inhibition of human PDE4A in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A

Assay data:46 Active, 10 Activity ≤ 1 µM, 927 Tested

AID:: 1961814

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196181310.

Compound was evaluated for inhibition of human PDE3A in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: cGMP-inhibited 3',5'-cyclic phosphodiesterase A

Assay data:15 Active, 6 Activity ≤ 1 µM, 927 Tested

AID:: 1961813

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196181211.

Binding affinity towards human OPRM1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Mu-type opioid receptor

Assay data:117 Active, 24 Activity ≤ 1 µM, 927 Tested

AID:: 1961812

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196178712.

Compound was evaluated for inhibition of human MAOA in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Amine oxidase [flavin-containing] A

Assay data:13 Active, 5 Activity ≤ 1 µM, 927 Tested

AID:: 1961787

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196178613.

Compound was evaluated for inhibition of human KDR in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: Vascular endothelial growth factor receptor 2

Assay data:19 Active, 11 Activity ≤ 1 µM, 692 Tested

AID:: 1961786

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196178514.

Compound was evaluated for inhibition of human KCNH2 in an in vitro assay with cellular components measured by membrane filtration, radioactivity method

Source:: ChEMBL

Protein Target:: Potassium voltage-gated channel subfamily H member 2

Assay data:353 Active, 116 Activity ≤ 1 µM, 1804 Tested

AID:: 1961785

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196177715.

Agonist activity at human HTR2B in an in vitro cell-based assay (CRO assay) measured by time-resolved fluorescence resonance energy transfer method

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2B

Assay data:3 Active, 5 Activity ≤ 1 µM, 927 Tested

AID:: 1961777

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196177216.

Binding affinity towards human HTR1A in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1A

Assay data:141 Active, 68 Activity ≤ 1 µM, 927 Tested

AID:: 1961772

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196176917.

Binding affinity towards human HRH3 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Histamine H3 receptor

Assay data:23 Active, 11 Activity ≤ 1 µM, 927 Tested

AID:: 1961769

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196175718.

Binding affinity towards rat Gabra1 in an in vitro assay with cellular components measured by scintillation counting

Source:: ChEMBL

Protein Target:: Gamma-aminobutyric acid receptor subunit alpha-1

Assay data:6 Active, 1 Activity ≤ 1 µM, 532 Tested

AID:: 1961757

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196175119.

Compound was evaluated for inhibition of human F2 in an in vitro cell free assay measured by fluorescence spectroscopy

Source:: ChEMBL

Protein Target:: Prothrombin

Assay data:11 Active, 8 Activity ≤ 1 µM, 927 Tested

AID:: 1961751

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 196174920.

Binding affinity towards human ESR1 in an in vitro cell free assay (CRO assay) measured by membrane filtration

Source:: ChEMBL

Protein Target:: Estrogen receptor

Assay data:31 Active, 1 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 927 Tested

AID:: 1961749

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Target

Proteins (200)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (330)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (70)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (241)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (294)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (21)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (146)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (40)
BioAssays extracted from the literature
NIH MLP (246)
BioAssays deposited by the NIH Molecular Libraries Program
Other (62)
BioAssays deposited by other experimentalists

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BioAssays for PubChem Compound (Select 2993) (350)
PubChem BioAssay
Nucleotide Links for Gene (Select 22911) (41)
Nucleotide
XM_006235063 (0)
GEO Profiles
WD repeat-containing protein 47 isoform X5 [Homo sapiens]
WD repeat-containing protein 47 isoform X5 [Homo sapiens]
gi|767903200|ref|XP_011539330.1|

Protein
WD repeat-containing protein 47 isoform X4 [Homo sapiens]
WD repeat-containing protein 47 isoform X4 [Homo sapiens]
gi|2462506298|ref|XP_054191181.1|

Protein

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