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GABAA (α1β2γ2) Receptor Current using Patch-Clamp Technique from US Patent US20240132445: "PHENOL DERIVATIVE AND APPLICATION THEREOF IN MEDICAMENTS"
Assay data:1 Active, 2 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Binding Assay from US Patent US20240067637: "NAPHTHYRIDINE AND PYRIDO[3,4-c]PYRIDAZINE DERIVATIVES AS GABAA ALPHA 5 RECEPTOR MODULATORS"
Assay data:44 Active, 1 Activity ≤ 1 nM, 44 Activity ≤ 1 µM, 44 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Patch Clamp Electrophysiology from US Patent US11912737: "19-nor neuroactive steroids and methods of use thereof"
Assay data:2 Active, 3 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
Steroid Inhibition of TBPS Binding from US Patent US11912737: "19-nor neuroactive steroids and methods of use thereof"
Assay data:4 Active, 47 Activity ≤ 1 µM, 47 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Binding Assay from US Patent US20240043418: "1,3-DIHYDRO-2H-PYRROLO[3,4-C]PYRIDINE DERIVATIVES AS GABAA A5 RECEPTOR MODULATORS"
Assay data:3 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
Cross screening panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
GABAA, Muscimol, Central Eurofins Panlabs panel
GABAA, Flunitrazepam, Central Eurofins Panlabs panel
GABAA, Chloride Channel, TBOB Eurofins Panlabs panel
BZD/CENTR/R Eurofins SafetyScreen44 (BI)
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