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Inhibition of P-gp (unknown origin) expressed in dog MDCK-MDR1cells assessed as maximum inhibition by calcein AM accumulation assay relative to control
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of P-gp (unknown origin) expressed in dog MDCK-MDR1cells assessed as maximum inhibition at 10 uM by calcein AM accumulation assay relative to control
Assay data:8 Tested
Inhibition of P-gp (unknown origin) at 10 uM incubated for 30 mins by calcein AM analysis relative to control
Assay data:34 Tested
Inhibition of P-gp (unknown origin) incubated for 30 mins by calcein AM analysis
Assay data:16 Active, 19 Tested
Inhibition of P-gp (unknown origin) expressed in dog MDCK-MDR1cells by calcein AM accumulation assay
Assay data:1 Active, 1 Tested
Inhibition of P-gp (unknown origin) expressed in human A2780 ADR cells by calcein AM accumulation assay
Inhibition of P-gp (unknown origin)
Assay data:6 Active, 2 Activity ≤ 1 µM, 7 Tested
Substrate activity at human P-gp assessed as efflux ratio
Substrate activity at human P-gp assessed as apparent permeability
Substrate activity at P-gp (unknown origin) expressed in MDCK-MDR1 cells assessed as efflux ratio by LC-MS/MS
Substrate activity at human P-gp in vinblastine-resistant human KBV cells overexpressing human tau protein assessed as efflux ratio
Assay data:33 Tested
Substrate activity at P-glycoprotein in human Caco-2 cells assessed as efflux ratio of permeability across basolateral to apical side over apical to basolateral side at 3 uM incubated for 2 hrs by LC-MS/MS analysis
Assay data:4 Tested
Binding affinity to P-gp in vincristine resistant human Eca-109 cells assessed as stabilization of protein at 67 degree C at 100 uM incubated for 30 mins by thermal shift assay
Assay data:2 Active, 2 Tested
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as increase in intracellular accumulation of calcein-AM at 1 to 5 uM incubated for 1 hr by flow cytometry analysis
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as increase in intracellular accumulation of rhodamine123 at 1 to 5 uM incubated for 1 hr by flow cytometry analysis
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as effect on accumulation of H33342
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as effect on accumulation of doxorubicin
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as effect on accumulation of calcein-AM
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as effect on accumulation of rhodamine123
Inhibition of P-gp efflux in vincristine resistant human Eca-109 cells assessed as increase in rhodamine 123 fluorescence intensity incubated for 3 hrs
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