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Selectivity interaction (KinomeScan (DiscoverX)) EUB0000304b TAOK3
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000306b TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000351a TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000710a TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000706a TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000702a TAOK1
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000305b TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000178b TAOK1
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000178b TAOK1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Enzymatic assay) EUB0000178b TAOK1
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000178b TAOK3
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000178b TAOK3
Selectivity interaction (Enzymatic assay) EUB0000178b TAOK3
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000178b TAOK2
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000178b TAOK2
Selectivity interaction (Enzymatic assay) EUB0000178b TAOK2
Inhibition of TAOK1 (unknown origin) at 0.1 uM relative to control
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of TAOK1 (unknown origin) at 1 uM relative to control
Inhibition of TAOK2 (TAO1) (unknown origin) at 1 uM relative to control
Inhibition of human partial length wild type TAOK1 by measuring selectivity score at 1 uM by Kinomescan method relative to control
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