Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Inhibition of EphA1 (unknown origin) at 1 uM relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000289c EPHA1
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000289c EPHA1
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000143b EPHA1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of EphA1 (unknown origin)
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
EPHA1 DiscoveRx kinase panel
EphA1(h) Kinase panel
EphA1(h) Millipore kinase panel
Inhibition of EPHA1 (unknown origin) at 1 uM
Inhibition of human recombinant EPHA1 incubated for 1 hrs by HTRF KinEASE TK assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Mobility Shift Assay from US Patent US9365572: "PI3K and/or mTOR inhibitor"
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
KinomeScan assay: inhibition of EPHA1
Assay data:108 Tested
EphA1(EPA1LGY1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
EphA1(h) Eurofins kinase panel
EPHA1 ProQinase selectivity panel
EPHA1 Kinase activity screen
EPHA1 Kinase screen
EPHA1 Invitrogen selectivity data (BI)
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on