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STLK5(STRAPHD1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of STLK5 in human NCI-H929 cells at 10 uM by mass spectroscopic analysis relative to control
Assay data:6 Tested
SummaryRelated BioAssays by Target
Inhibition of STLK5 in human NCI-H929 cells by mass spectroscopic analysis
Assay data:2 Active, 6 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Binding affinity to LYK5 in human SUM159 cell lysates by multiplexed inhibitor bead profiling-based LC-MS/MS analysis
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of STLK5 in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled YSVKVLPWLSPEVLQQNLQGYDAK probe by mass-spectrometric analysis relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of STLK5 activation loop (unknown origin) at 10 uM
Assay data:1 Tested
Inhibition of recombinant full-length N-terminal 6-His-tagged human LKB1/GST-tagged MO25alpha/GST-tagged STRADalpha expressed in SF21 cells at 3 uM relative to control
Inhibition of STLK5 conserved Lys2 (SVKASHILISVDGK) in human PBMC at 0.1 uM
Inhibition of STLK5 activation loop (YSVKVLPWLSPEVLQQNLQGYDAK) in human PBMC at 0.1 uM
Inhibition of STLK5 conserved Lys2 (SVKASHILISVDGK) in human PBMC at 1 uM
Inhibition of STLK5 activation loop (YSVKVLPWLSPEVLQQNLQGYDAK) in human PBMC at 1 uM
Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.
Assay data:5 Active, 2 Activity ≤ 1 µM, 237 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of LKB1-MO25a-STRADa at 10 uM
Inhibition of human STLK5 in HL-60 cells lysate assessed as reduction of labeling of acyl-phosphate ATP probe at 100 nM
Assay data:4 Tested
Inhibition of human STLK5 in HL60 cells lysate at 10 uM using post probe-labeling by LC-MS/MS analysis relative to control
Assay data:5 Tested
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