Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Inhibition of Bub1 (unknown origin) by bio-chip based analysis
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000309b BUB1
SummaryRelated BioAssays by Target
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000540a BUB1
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000335a BUB1
BUB1 DiscoveRx kinase panel
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Abrogation of histone H2A-Thr120 phosphorylation
TR-FRET
ePCA binding competition (equilibrium binding assay)
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
BUB1 surface plasmon resonance (SPR) assay
BUB1 biochemical assay (high ATP)
Assay data:2 Tested
BUB1 biochemical assay (low ATP)
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Kinase Assay from US Patent US10428063: "4H-pyrrolo[3,2-C]pyridin-4-one derivatives"
Assay data:46 Active, 46 Activity ≤ 1 µM, 46 Tested
Kinase Assay from US Patent US10428044: "3-amino-1,5,6,7-tetrahydro-4H-indol-4-ones"
Assay data:466 Active, 404 Activity ≤ 1 µM, 480 Tested
Bub1 Kinase Assay from US Patent US10308629: "1H-pyrrol-3-amines"
Assay data:40 Active, 39 Activity ≤ 1 µM, 40 Tested
Bub1 Kinase Assay from US Patent US10266548: "Substituted benzylindazoles for use as Bub1 kinase inhibitors in the treatment of hyperproliferative diseases"
Assay data:183 Active, 159 Activity ≤ 1 µM, 187 Tested
Bub1 kinase assay from US Patent US10227299: "3-amino-1,5,6,7-tetrahydro-4H-indol-4-ones"
Assay data:287 Active, 280 Activity ≤ 1 µM, 287 Tested
Time-Resolved Fluorescence Energy Transfer (TR-FRET) Kinase Assay from US Patent US9765058: "Substituted benzylpyrazoles"
Assay data:19 Active, 18 Activity ≤ 1 µM, 19 Tested
Bub1 Kinase Assay from US Patent US9682995: "Amino-substituted isothiazoles"
Assay data:6 Active, 1 Activity ≤ 1 µM, 121 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
KinomeScan assay: inhibition of BUB1
Assay data:3 Active, 108 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Bub1(BUB1LGRL) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on