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Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranes
Assay data:7 Active, 4 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at human recombinant sst1 receptor assessed as inhibition of SRIF28-induced luciferase activity
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Antagonist activity at human recombinant sst1 receptor in CCl39 cells assessed as SRIF14-induced inhibition of forskolin-stimulated adenylate cyclase activity
Binding affinity to human recombinant sst1 receptor
Assay data:4 Active, 3 Activity ≤ 1 µM, 4 Tested
Displacement of [125I](Leu8,D-Trp22,Tyr25)-SRIF28 from human sst1 receptor
Assay data:2 Active, 4 Activity ≤ 1 µM, 4 Tested
Antagonist activity at human recombinant sst1 receptor assessed as blockade of SRIF14-induced inhibition of forskolin stimulated adenylate cyclase activity
Assay data:1 Tested
Assay data:1 Active, 1 Activity ≤ 1 µM, 3 Tested
Binding affinity to human SST1R
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptor
Displacement of [125I][LTT]SRIF28 from human cloned sst1 receptor by autoradiography
Assay data:1 Active, 33 Activity ≤ 1 µM, 33 Tested
Affinity for somatostatin receptors
Inhibition of sst receptor at 10 uM
Inhibition of sst receptor at 1 uM
Inhibition of [125I](Leu8,DTrp22,Tyr25)-SRIF28 binding to human sst1
Assay data:6 Activity ≤ 1 µM, 6 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to somatostatin receptor by radioligand binding assay
Binding affinity for SRIF (somatostatin) receptor
Assay data:5 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 11 Tested
Binding affinity towards somatostatin receptor type 1
Assay data:2 Active, 3 Activity ≤ 1 µM, 3 Tested
In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 1 expressed in CHO-K1 cells; (n=7)
Binding affinity to human sst1 receptor expressed in Chinese hamster CCL39 cells by autoradiography
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