Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Safety47 Scan (DiscoverX - Eurofins)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Uptake, Dopamine - Antagonist Eurofins Panlabs panel
Transporter, Dopamine (DAT) Eurofins Panlabs panel
DATRANS/HUM Eurofins SafetyScreen44 (BI)
Binding affinity towards human SLC6A3 in an in vitro assay with cellular components measured by scintillation counting
Assay data:119 Active, 21 Activity ≤ 1 µM, 1213 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Assay data:128 Active, 38 Activity ≤ 1 µM, 927 Tested
Displacement of [3H]nisoxetine from recombinant human Dopamine transporter at 10 uM after 120 mins by scintillation counting analysis relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of dopamine transporter (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of DAT (unknown origin) at 10 uM
Inhibition of dopamine transporter (unknown origin) assessed as inhibition of dopamine reuptake
Assay data:5 Active, 3 Activity ≤ 1 µM, 5 Tested
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000295b SLC6A3
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (GPCR panel (PDSP screen)) EUB0000545a SLC6A3
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Lead profiling screen (Eurofins, GPCRs, ion channels, kinases and transporters)) EUB0000309b SLC6A3
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on