BioAssay by Target (List) for Gene (Select 5585) - PubChem BioAssay - NCBI

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Select item 18791321.

Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:9 Active, 5 Activity ≤ 1 µM, 15 Tested

AID:: 1879132

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18791312.

Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysis

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:9 Active, 7 Activity ≤ 1 µM, 15 Tested

AID:: 1879131

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18355923.

PKN1 DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1835592

Summary Related BioAssays by Target

Select item 18351294.

PRK1(h) Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1835129

Summary Related BioAssays by Target

Select item 18342955.

Inhibition of PKN1 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1834295

Summary PubMed Citation Related BioAssays by Target

Select item 17942846.

KinomeScan assay: inhibition of PKN1

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:108 Tested

AID:: 1794284

Summary Related BioAssays by Target

Select item 17937737.

PKN1 [PRK1(PKN1LGY1)] Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793773

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17934868.

PKN1 [PRK1(PKN1LGY1)] Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793486

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17931929.

PKN1 [PRK1(PKN1LGY1)] Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793192

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179282510.

PRK1(h) Eurofins kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1792825

Summary Related BioAssays by Target

Select item 179243611.

PRK1 ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1792436

Summary Related BioAssays by Target

Select item 179114012.

PKN1 (PRK1) Kinase screen

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1791140

Summary Related BioAssays by Target

Select item 179031913.

PKN1 Invitrogen selectivity data (BI)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1790319

Summary Related BioAssays by Target

Select item 178943214.

PRK1(h) Eurofins Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1789432

Summary Related BioAssays by Target

Select item 178766015.

PKN1 (PRK1) SelectScreen Kinase panel (LifeTechnologies)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1787660

Summary Related BioAssays by Target

Select item 178748616.

PRK1(h) Millipore kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1787486

Summary Related BioAssays by Target

Select item 178651417.

PKN1 Invitrogen Lab (UK) kinase screen (BI)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1786514

Summary Related BioAssays by Target

Select item 178605318.

PRK1 Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1786053

Summary Related BioAssays by Target

Select item 176803919.

Inhibition of PAK1 transcriptional activity in human KMS-11 cells assessed as reduction in H3K36 methylation at 10 uM measured after 72 hrs by chip q-PCR analysis

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Active, 1 Tested

AID:: 1768039

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 175345920.

Inhibition of full length N-terminal GST-tagged PAK1 (1 to 545 residues) (unknown origin) expressed in Sf21 at 10 uM preincubated for 10 mins followed by peptide substrate addition relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N1

Assay data:1 Tested

AID:: 1753459

Summary PubMed Citation Related BioAssays by Target

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Target

Proteins (3)
BioAssays with protein sequences specified as targets
RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (31)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (3)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (23)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (36)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (139)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (44)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (1)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (111)
BioAssays extracted from the literature
NIH MLP (2)
BioAssays deposited by the NIH Molecular Libraries Program
Other (69)
BioAssays deposited by other experimentalists

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BioAssay by Target (List) for Gene (Select 5585) (183)
PubChem BioAssay
dbVar for Gene (Select 5585) (268)
dbVar
PKN1[gene] (99)
ClinVar
RecName: Full=Protein FAM177B
RecName: Full=Protein FAM177B
gi|172048722|sp|A6PVY3.1|F177B_HUMA

Protein

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