BioAssay by Target (List) for Gene (Select 5142) - PubChem BioAssay - NCBI

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Select item 19636111.

Biochemical Kinase Assay Protocol (JAK) from US Patent US20240132525: "BORON CONTAINING PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM, METHODS AND USES THEREOF"

Source:: BindingDB

Protein Targets:: Tyrosine-protein kinase JAK1; ...
Total:: 3

Assay data:90 Active, 39 Activity ≤ 1 nM, 91 Activity ≤ 1 µM, 91 Tested

AID:: 1963611

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19635162.

In vitro PDE4B Enzyme Activity Detection Assay from US Patent US20240083921: "BORATE DERIVATIVE AND USES THEREOF"

Source:: BindingDB

Protein Targets:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B; ...
Total:: 1

Assay data:14 Active, 12 Activity ≤ 1 nM, 14 Activity ≤ 1 µM, 14 Tested

AID:: 1963516

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19632663.

Cross screening panel

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1963266

Summary Related BioAssays by Target

Select item 19632174.

Cross screening panel

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1963217

Summary Related BioAssays by Target

Select item 19631675.

Cross screening panel

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1963167

Summary Related BioAssays by Target

Select item 19624976.

Phosphodiesterase PDE4 Eurofins Panlabs panel

Source:: ChEMBL

Protein Targets:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A; ...
Total:: 4

Assay data:1 Tested

AID:: 1962497

Summary Related BioAssays by Target

Select item 19624717.

Panlabs assay PDE4B1

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1962471

Summary Related BioAssays by Target

Select item 19624588.

3H-cAMP and 3H-cGMP Scintillation Proximity Assay (PDE4B)

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1962458

Summary Related BioAssays by Target

Select item 19612569.

Inhibition of PDE4B (unknown origin) upto 10000 nM

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1961256

Summary PubMed Citation Related BioAssays by Target

Select item 196069110.

Inhibition of PDE4B (unknown origin) by 3H-cAMP scintillation proximity assay

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1960691

Summary PubMed Citation Related BioAssays by Target

Select item 193410111.

Inhibition of human recombinant PDE4B incubated for 30 mins by Scintillation Proximity Assay

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1934101

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 193332012.

Inhibition of human recombinant PDE4B

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:4 Active, 1 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 4 Tested

AID:: 1933320

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192953513.

Inhibition of human PDE4 catalytic domain expressed in Escherichia coli at 10 uM relative to control

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Tested

AID:: 1929535

Summary PubMed Citation Related BioAssays by Target

Select item 192953414.

Inhibition of human PDE4 catalytic domain expressed in Escherichia coli

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:10 Active, 5 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 12 Tested

AID:: 1929534

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192445415.

Binding affinity to human PDE4 assessed as dissociation constant

Source:: ChEMBL

Protein Targets:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A; ...
Total:: 4

Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1924454

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192444916.

Inhibition of human PDE4

Source:: ChEMBL

Protein Targets:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A; ...
Total:: 4

Assay data:1 Tested

AID:: 1924449

Summary PubMed Citation Related BioAssays by Target

Select item 192356217.

Inhibition of human recombinant PDE4B1 using FAM-cAMP as substrate incubated for 20 mins

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1923562

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192356018.

Displacement of [3H]-cAMP from full-length recombinant human PDE4B1 by fluorescence polarisation assay

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1923560

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192355919.

Inhibition of PDE4B (unknown origin)

Source:: ChEMBL

Protein Target:: cAMP-specific 3',5'-cyclic phosphodiesterase 4B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1923559

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192355820.

Inhibition of PDE4 (unknown origin)

Source:: ChEMBL

Protein Targets:: cAMP-specific 3',5'-cyclic phosphodiesterase 4A; ...
Total:: 4

Assay data:3 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1923558

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Activity (IC50, etc) ≤ 1 nM (115)
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Activity (IC50, etc) ≤ 1 µM (377)
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Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
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BioAssay by Target (List) for Gene (Select 5142) (717)
PubChem BioAssay
Maged1 MAGE family member D1 [Mus musculus]
Maged1 MAGE family member D1 [Mus musculus]
Gene ID:94275

Gene
94275[uid] AND (alive[prop]) (1)
Gene

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