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In Vitro Radioligand Binding Assay from US Patent US20240208984: "BIVALENT LIGANDS TO UNDERSTAND DIMERIZATION OF THE MU OPIOID RECEPTOR AND THE CHEMOKINE RECEPTOR CCR5 IN NEUROLOGICAL DISORDERS"
Assay data:6 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 6 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibitory Effects on Recombinant AOX Protein from US Patent US11565996: "Compounds for use as inhibitors of alternative oxidase or cytochrome bc1 complex"
Assay data:4 Active, 3 Activity ≤ 1 µM, 4 Tested
beta-lactamase assay from US Patent US10543221: "Beta-lactamase inhibitors, formulations, and uses thereof"
Assay data:6 Active, 1 Activity ≤ 1 µM, 13 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Stopped Flow CO2 Hydration Assay from Article 10.3109/14756366.2013.813942: "Biochemical characterization of the chloroplastic -carbonic anhydrase from Flaveria bidentis (L.) "Kuntze"."
Assay data:14 Tested
SummaryPubMed CitationRelated BioAssays by Target
Urease Inhibition Assay from Article 10.3109/14756366.2012.740477: "Synthesis and biological evaluation of novel series of aminopyrimidine derivatives as urease inhibitors and antimicrobial agents."
Assay data:17 Tested
Inhibition Assay from US Patent US9447057: "Schiff bases of thiazoles: a new class of ureases inhibitors"
Assay data:9 Active, 29 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Kinetic Assay from Article 10.3109/14756366.2012.668539: "Inhibition of cysteine proteases by a natural biflavone: behavioral evaluation of fukugetin as papain and cruzain inhibitor."
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
In Vitro LOX Inhibition Assay from Article 10.3109/14756366.2011.555944: "Synthesis and biological evaluation of fused oxepinocoumarins as free radicals scavengers."
Assay data:3 Tested
LOX Activity Assay from Article 10.3109/14756366.2010.529807: "Inhibition of lipoxygenase (LOX) and anticancer activity caused by gold(I) mixed ligands complexes of triphenylphosphine and thioamides."
Assay data:1 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Urease Inhibition Assay from Article 10.3109/14756366.2010.528415: "Urease inhibitors from Indigofera gerardiana Wall."
Lipoxygenase Activity Assay from Article 10.3109/14756366.2010.495717: "Synthesis and SAR comparative studies of 2-allyl-4-methoxy-1-alkoxybenzenes as 15-lipoxygenase inhibitors."
Assay data:4 Active, 13 Tested
SummaryCompounds, ActivePubMed Citation
Urease Inhibition Assay from Article 10.3109/14756360903389864: "Design, synthesis, and urease inhibition studies of some 1,3,4-oxadiazoles and 1,2,4-triazoles derived from mandelic acid."
Assay data:7 Tested
Urease Inhibition Assay from Article 10.3109/14756360903179385: "Urease inhibitors from Hypericum oblongifolium WALL."
Assay data:4 Tested
Lipoxygenase Inhibition Assay from Article 10.1080/14756360903179484: "Conferin, potent antioxidant and anti-inflammatory isoflavone from Caragana conferta Benth."
In Vitro Soybean Lipoxygenase (SLO) Inhibition Assay from Article 10.1016/j.bioorg.2017.01.016: "Substituted furans as potent lipoxygenase inhibitors: Synthesis, in vitro and molecular docking studies."
Assay data:11 Tested
SummaryPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Isothermal Titration Calorimetry (ITC) from Article 10.1074/jbc.M113.487777: "Roles of phosphate recognition in inositol 1,3,4,5,6-pentakisphosphate 2-kinase (IPK1) substrate binding and activation."
Assay data:3 Active, 1 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Lipo-oxygenase Inhibitory Assay from Article 10.1111/cbdd.12779: "2-Prenylated m-dimethoxybenzenes as potent inhibitors of 15-lipo-oxygenase: inhibitory mechanism and SAR studies."
Assay data:3 Active, 1 Activity ≤ 1 µM, 11 Tested
Urease Inhibition Assay from Article 10.1016/j.bioorg.2016.03.010: "Hybrid benzothiazole analogs as antiurease agent: Synthesis and molecular docking studies."
Assay data:11 Active, 21 Tested
Urease Inhibition Assay from Article 10.1111/cbdd.12675: "Iminothiazoline-Sulfonamide Hybrids as Jack Bean Urease Inhibitors; Synthesis, Kinetic Mechanism and Computational Molecular Modeling."
Assay data:10 Active, 10 Activity ≤ 1 µM, 11 Tested
Urease Inhibition Assay from Article 10.1016/j.bioorg.2015.12.007: "Dihydropyrimidine based hydrazine dihydrochloride derivatives as potent urease inhibitors."
Assay data:13 Tested
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