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Competition Binding Assay from US Patent US20240293587: "CXCR4-TARGETED DIAGNOSTIC AND THERAPEUTIC AGENTS WITH REDUCED SPECIES SELECTIVITY"
Assay data:29 Active, 1 Activity ≤ 1 nM, 30 Activity ≤ 1 µM, 30 Tested
SummaryRelated BioAssays by Target
Receptor Binding Assay from US Patent USRE48059: "Piperazine-substituted benzothiophenes for treatment of mental disorders"
Assay data:59 Active, 2 Activity ≤ 1 nM, 59 Activity ≤ 1 µM, 59 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Assay data:57 Active, 18 Activity ≤ 1 nM, 57 Activity ≤ 1 µM, 57 Tested
Cell based assay rat (ADRA2B)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of Transporter, GABA at 10.0 M in the Eurofins Panlabs Safety Screen
Assay data:1 Tested
Inhibition of Purinergic P2Y, non-selective at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of Purinergic P2X at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of Glutamate, NMDA, Glycine at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of Glutamate, NMDA, Agonism at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of GABAB, Non-Selective at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of GABAA, Flunitrazepam, Central at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of GABAA, Chloride Channel, TBOB at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of Adrenergic alpha1A at 10.0 M in the Eurofins Panlabs Safety Screen
Inhibition of Aldose Reductase at 10.0 M in the Eurofins Panlabs Safety Screen
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