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Radioligand Binding Assay on Mouse TAAR1 from US Patent US11697636: "Substituted benzamides"
Assay data:298 Active, 20 Activity ≤ 1 nM, 279 Activity ≤ 1 µM, 300 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Enzymatic Assay for MASP-2 from US Patent US11584714: "MASP-2 inhibitors and methods of use"
Assay data:436 Active, 324 Activity ≤ 1 µM, 479 Tested
Biological Assay (RFMS) from US Patent US11198681: "Heteroaryl inhibitors of PAD4"
Assay data:43 Active, 11 Activity ≤ 1 µM, 80 Tested
Receptor [35S] GTPgammaS Binding Assays: (S1P1 GTPgammaS/S1P3 GTPgammaS) from US Patent US11058696: "Substituted bicyclic compounds"
Assay data:12 Active, 1 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 12 Tested
S1P1 Binding Assay from US Patent US11058696: "Substituted bicyclic compounds"
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
STING SPA Binding Assay from US Patent US11021511: "Cyclic dinucleotides as sting agonists"
Assay data:5 Active, 5 Activity ≤ 1 µM, 6 Tested
FLIPR and cAMP Inhibition Assay from US Patent US10858365: "Triazolo-pyrimidine compounds and uses thereof"
Assay data:117 Active, 13 Activity ≤ 1 nM, 116 Activity ≤ 1 µM, 119 Tested
Enzymatic Activity Assay of MetAP2 from US Patent US10807971: "Pyrrolidinone compounds"
Assay data:17 Active, 17 Activity ≤ 1 µM, 17 Tested
Enzymatic Activity Assay of DPP-4 from US Patent US10807971: "Pyrrolidinone compounds"
Assay data:17 Active, 3 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 17 Tested
Enzyme Inhibition Assay from US Patent US10759791: "Mammalian and bacterial nitric oxide synthase inhibitors"
Assay data:24 Active, 21 Activity ≤ 1 µM, 24 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Caliper Kinase Assay from US Patent US10676460: "Quinazolines as potassium ion channel inhibitors"
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding Assays from US Patent US10577368: "A3 adenosine receptor agonists"
Assay data:61 Active, 18 Activity ≤ 1 nM, 61 Activity ≤ 1 µM, 61 Tested
Radioligand Binding Assay from US Patent US9452980: "Substituted benzamides"
Assay data:301 Active, 20 Activity ≤ 1 nM, 282 Activity ≤ 1 µM, 302 Tested
In Vitro Cell Proliferation Potency Assay from US Patent US9434725: "5-azaindazole compounds and methods of use"
Assay data:109 Active, 70 Activity ≤ 1 µM, 110 Tested
Competition Receptor Binding Assay from US Patent US9416103: "Use of the aminoalkylindole JWH-073-M4 and related compounds as neutral CB1 receptor antagonists for the treatment of alcoholism, drug abuse, obesity, and obesity-related diseases"
Assay data:6 Active, 1 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 6 Tested
Fluorescence Polarization Assay (FPA) from US Patent US9345740: "IAP antagonists"
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
SelectScreen Biochemical Kinase Assay from Article 10.1074/jbc.M113.507525: "Effects of isoform-selective phosphatidylinositol 3-kinase inhibitors on osteoclasts: actions on cytoskeletal organization, survival, and resorption."
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition Assay from US Patent US9271969: "Compounds as inhibitors of diacylglycerol O-acyltransferase type 1 enzyme"
Assay data:67 Active, 8 Activity ≤ 1 nM, 67 Activity ≤ 1 µM, 67 Tested
Endothelial Lipase Assay from US Patent US9216998: "Tricyclic indole derivatives useful endothelial lipase inhibitors"
Assay data:26 Active, 24 Activity ≤ 1 µM, 27 Tested
Inhibition Assay from US Patent US9181187: "Therapeutic agent for urinary excretion disorder"
Assay data:12 Active, 12 Activity ≤ 1 µM, 12 Tested
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