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Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.
Figure 3Modifications to the isatin core of ML129
- PMCPubMed Central citations
- PubChem BioAssay for Chemical ProbePubChem BioAssay records reporting screening data for the development of the chemical probe(s) described in this book chapter
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- Review Development of the First CNS penetrant M5 Positive Allosteric Modulator (PAM) Based on a Novel, non-Isatin Core.[Probe Reports from the NIH Mol...]Review Development of the First CNS penetrant M5 Positive Allosteric Modulator (PAM) Based on a Novel, non-Isatin Core.Gentry PR, Kokubo M, Bridges TM, Daniels JS, Niswender CM, Smith E, Chase P, Hodder PS, Rosen H, Conn PJ, et al. Probe Reports from the NIH Molecular Libraries Program. 2010
- Discovery of ML326: The first sub-micromolar, selective M5 PAM.[Bioorg Med Chem Lett. 2013]Discovery of ML326: The first sub-micromolar, selective M5 PAM.Gentry PR, Bridges TM, Lamsal A, Vinson PN, Smith E, Chase P, Hodder PS, Engers JL, Niswender CM, Daniels JS, et al. Bioorg Med Chem Lett. 2013 May 15; 23(10):2996-3000. Epub 2013 Mar 16.
- Review Development of the First Potent, Selective and CNS penetrant M5 Negative Allosteric Modulator (NAM).[Probe Reports from the NIH Mol...]Review Development of the First Potent, Selective and CNS penetrant M5 Negative Allosteric Modulator (NAM).Gentry PR, Kokubo M, Bridges TM, Daniels JS, Niswender CM, Smith E, Chase P, Hodder PS, Rosen H, Conn PJ, et al. Probe Reports from the NIH Molecular Libraries Program. 2010
- Review Development of a Novel, Orthosteric M5 Antagonist Possessing a High Degree of Muscarinic Subtype Selectivity.[Probe Reports from the NIH Mol...]Review Development of a Novel, Orthosteric M5 Antagonist Possessing a High Degree of Muscarinic Subtype Selectivity.Gentry PR, Kokubo M, Bridges TM, Daniels JS, Niswender CM, Smith E, Chase P, Hodder PS, Rosen H, Conn PJ, et al. Probe Reports from the NIH Molecular Libraries Program. 2010
- Review Development of the First Highly Selective mAChR 5 (M(5)) Positive Allosteric Modulator (PAM).[Probe Reports from the NIH Mol...]Review Development of the First Highly Selective mAChR 5 (M(5)) Positive Allosteric Modulator (PAM).Bridges TM, Lewis LM, Weaver CD, Wood MR, Daniels JS, Conn PJ, Lindsley CW. Probe Reports from the NIH Molecular Libraries Program. 2010
- Figure 3, Modifications to the isatin core of ML129 - Probe Reports from the NIH...Figure 3, Modifications to the isatin core of ML129 - Probe Reports from the NIH Molecular Libraries Program
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