A New Nucleoside Antibiotic Chokes Bacterial RNA Polymerase

Biochemistry. 2017 Sep 19;56(37):4923-4924. doi: 10.1021/acs.biochem.7b00680. Epub 2017 Sep 8.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / pharmacology*
  • DNA-Directed RNA Polymerases / antagonists & inhibitors*
  • Enzyme Inhibitors / pharmacology*
  • Humans
  • Methicillin-Resistant Staphylococcus aureus / drug effects
  • Methicillin-Resistant Staphylococcus aureus / enzymology
  • Mice
  • Nucleosides / pharmacology*
  • Streptococcus pneumoniae / drug effects
  • Streptococcus pneumoniae / enzymology

Substances

  • Anti-Bacterial Agents
  • Enzyme Inhibitors
  • Nucleosides
  • DNA-Directed RNA Polymerases