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WHO-TDR: Lymphatic Filariasis
Assay data:76 Tested
Summary
Toxicity in Brugia malayi infected with Wolbachia assessed as decrease in microfilaria motility at 5 uM measured after 6 days
Assay data:1 Tested
SummaryPubMed Citation
Competitive inhibition of Brugia malayi T6PP using T6P as substrate by Lineweaver-Burk plot analysis
Assay data:1 Active, 7 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of sodium arsenate activated N-terminal GST-tagged Brugia malayi MPK1 expressed in HEK293F cells using FAM-p38tide as substrate by IMAP assay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Inhibition of recombinant Brugia malayi MPK1a using FAM-p38tide as substrate by IMAP assay
Assay data:8 Active, 8 Activity ≤ 1 µM, 8 Tested
Antifilarial activity against Brugia malayi microfilariae isolated from peritoneal cavity of infected Meriones unguiculatus assessed as loss of motility incubated for 48 hrs by microscopy
Assay data:5 Active, 13 Tested
SummaryCompounds, ActivePubMed Citation
AntiBrugia malayi activity Effect on motility
Assay data:1 Active, 2 Tested
SummaryCompounds, Active
Inhibition of recombinant Brugia malayi DPY-31 astacin domain expressed in Escherichia coli using Suc-Ala-Ala-Ala-pNA as substrate preincubated for 3 hrs followed by substrate addition measured after 3 hrs by microplate reader assay
Assay data:5 Tested
SummaryPubMed CitationRelated BioAssays by Target
Antifilarial activity against Brugia malayi microfilariae assessed as motility reduction after 1 hr by microscopic analysis
Assay data:3 Active, 3 Tested
Antifilarial activity against adult Brugia malayi assessed as motility reduction after 1 hr by microscopic analysis
Inhibition of recombinant Brugia malayi TMK using dTMP as substrate by pyruvate kinase/lactate dehydrogenase coupled assay
Assay data:7 Active, 15 Tested
Antifilarial activity against Brugia malayi microfilaria assessed as reduction in motility after 5 days by MTT dye reduction assay
Assay data:8 Active, 7 Activity ≤ 1 µM, 12 Tested
Antifilarial activity against Brugia malayi adult worm assessed as reduction in motility after 5 days by MTT dye reduction assay
Assay data:8 Active, 5 Activity ≤ 1 µM, 12 Tested
Inhibition of Brugia malayi thymidylate kinase using dTMP substrate by spectrophotometric assay
Assay data:3 Active, 15 Tested
Antifilarial activity against Brugia malayi microflilariae worm assessed as inhibition of parasite motility after 48 hrs by microscopic analysis
Assay data:4 Active, 16 Tested
Antifilarial activity against Brugia malayi adult worm assessed as inhibition of parasite motility after 48 hrs by microscopic analysis
Assay data:3 Active, 1 Activity ≤ 1 µM, 16 Tested
Antifilarial activity against female adult Brugia malayi assessed as inhibition of motility after 24 hrs by microscopic analysis
Assay data:1 Active, 8 Tested
Antifilarial activity against microfilariae Brugia malayi assessed as inhibition of motility after 24 hrs by microscopic analysis
Assay data:4 Active, 8 Tested
Assay data:8 Active, 3 Activity ≤ 1 µM, 8 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Assay data:52 Active, 1 Activity ≤ 1 µM, 52 Tested
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