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Antimicrobial Susceptibility Testing Assay from US Patent US10030047: "Peptide macrocycles against acinetobacter baumannii"
Assay data:50 Active, 35 Activity ≤ 1 µM, 55 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibition of carbapenem-resistant Acinetobacter baumannii ATCC 17978 OXA-24/40 expressed in Escherichia coli BL21 using nitrocefin as substrate measured after 15 mins by spectrophotometry analysis
Assay data:6 Active, 6 Activity ≤ 1 µM, 7 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Antibacterial activity against Acinetobacter baumannii ATCC 17978 transfected with pNT255:ADC-1 after 18 hrs by broth microdilution method
Assay data:1 Active, 7 Tested
SummaryCompounds, ActivePubMed Citation
Antibacterial activity against Acinetobacter baumannii ATCC 17978 transfected with pNT255 after 18 hrs by broth microdilution method
Assay data:2 Active, 2 Activity ≤ 1 µM, 7 Tested
Antibacterial activity against Acinetobacter baumannii ATCC 17978 after 18 hrs by broth microdilution method
Antibacterial activity against Acinetobacter baumannii ATCC 17978 col10 after 18 hrs by broth microdilution method
Assay data:15 Active, 9 Activity ≤ 1 µM, 16 Tested
Assay data:13 Active, 3 Activity ≤ 1 µM, 16 Tested
Antimicrobial activity against Acinetobacter baumannii ATCC 17978 incubated overnight by microdilution method
Assay data:7 Active, 19 Tested
Antibacterial activity against Acinetobacter baumannii ATCC 17978 after overnight incubation by microplate checkerbroad assay in presence of PSPC
Assay data:1 Tested
SummaryPubMed Citation
Inhibition of OXA-23 in carbapenem-resistant Acinetobacter baumannii ATCC 17978 transfected with pET-RA-KmR plasmid encoding rifampicin and kanamycin resistance assessed as potentiation of imipenem-induced antibacterial activity by measuring imipenem MIC at 16 ug/mL in Mueller-Hinton broth by CLSI protocol based method (Rvb = 8 ug/mL)
Assay data:9 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of OXA-24/40 in carbapenem-resistant Acinetobacter baumannii ATCC 17978 transfected with pET-RA-KmR plasmid encoding rifampicin and kanamycin resistance assessed as potentiation of imipenem-induced antibacterial activity by measuring imipenem MIC at 16 ug/mL in Mueller-Hinton broth by CLSI protocol based method (Rvb = 64 ug/mL)
Binding affinity to OXA-24/40 in carbapenem-resistant Acinetobacter baumannii ATCC 17978 assessed as ezyme-compound adduct formation from loss of catechol group with increase in mass at 1:100 ezyme-compound ratio using nitrocefin as substrate at pH 7 and 25 degree C by MALDI-TOF MS analysis
Assay data:3 Active, 3 Tested
Inhibition of carbapenem-resistant Acinetobacter baumannii ATCC 17978 OXA-24/40 expressed in Escherichia coli BL21 using nitrocefin as substrate measured after 15 mins by spectrophotometry analysis relative to parent compound
Inhibition of carbapenem-resistant Acinetobacter baumannii ATCC 17978 OXA-24/40 expressed in Escherichia coli BL21 assessed as ratio of Kinact/Ki using nitrocefin as substrate measured after 15 mins by spectrophotometry analysis relative to parent compound
Inhibition of Acinetobacter baumannii ATCC 17978 OXA-24/40 expressed in Escherichia coli BL21 assessed as ratio of Kinact/Ki using nitrocefin as substrate measured after 15 mins by spectrophotometry analysis
Assay data:7 Tested
Inhibition of carbapenem-resistant Acinetobacter baumannii ATCC 17978 OXA-24/40 expressed in Escherichia coli BL21 assessed as inactivation rate constant using nitrocefin as substrate measured after 15 mins by spectrophotometry analysis
Antibacterial activity against Acinetobacter baumannii ATCC 17978 harboring pAB880
Assay data:2 Tested
Antibacterial activity against Acinetobacter baumannii ATCC 17978
Antibacterial activity against Acinetobacter baumannii ATCC 17978 harboring plasmid directed expression of beta-lactamase OXA-58 under an ISAba3 promoter
Antibacterial activity against Acinetobacter baumannii ATCC 17978 harboring plasmid 1266
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