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Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.
Figure 7Validated hit resulting from the preliminary commercial SAR effort
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- A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry.[J Biomol Screen. 2013]A selective ATP-binding cassette subfamily G member 2 efflux inhibitor revealed via high-throughput flow cytometry.Strouse JJ, Ivnitski-Steele I, Khawaja HM, Perez D, Ricci J, Yao T, Weiner WS, Schroeder CE, Simpson DS, Maki BE, et al. J Biomol Screen. 2013 Jan; 18(1):26-38. Epub 2012 Aug 24.
- Grid-independent Descriptors (GRIND) Analysis and SAR Guided Molecular Docking Studies to Probe Selectivity Profiles of Inhibitors of Multidrug Resistance Transporters ABCB1 and ABCG2.[Curr Cancer Drug Targets. 2017]Grid-independent Descriptors (GRIND) Analysis and SAR Guided Molecular Docking Studies to Probe Selectivity Profiles of Inhibitors of Multidrug Resistance Transporters ABCB1 and ABCG2.Shafi T, Jabeen I. Curr Cancer Drug Targets. 2017; 17(2):177-190.
- Dacomitinib antagonizes multidrug resistance (MDR) in cancer cells by inhibiting the efflux activity of ABCB1 and ABCG2 transporters.[Cancer Lett. 2018]Dacomitinib antagonizes multidrug resistance (MDR) in cancer cells by inhibiting the efflux activity of ABCB1 and ABCG2 transporters.Fan YF, Zhang W, Zeng L, Lei ZN, Cai CY, Gupta P, Yang DH, Cui Q, Qin ZD, Chen ZS, et al. Cancer Lett. 2018 May 1; 421:186-198. Epub 2018 Jan 11.
- Review The role of multidrug resistance efflux transporters in antifolate resistance and folate homeostasis.[Drug Resist Updat. 2006]Review The role of multidrug resistance efflux transporters in antifolate resistance and folate homeostasis.Assaraf YG. Drug Resist Updat. 2006 Aug-Oct; 9(4-5):227-46. Epub 2006 Nov 7.
- Review Multidrug resistance proteins: role of P-glycoprotein, MRP1, MRP2, and BCRP (ABCG2) in tissue defense.[Toxicol Appl Pharmacol. 2005]Review Multidrug resistance proteins: role of P-glycoprotein, MRP1, MRP2, and BCRP (ABCG2) in tissue defense.Leslie EM, Deeley RG, Cole SP. Toxicol Appl Pharmacol. 2005 May 1; 204(3):216-37.
- Figure 7, Validated hit resulting from the preliminary commercial SAR effort - P...Figure 7, Validated hit resulting from the preliminary commercial SAR effort - Probe Reports from the NIH Molecular Libraries Program
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